Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50000864
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262192(CHEMBL4083840)
Affinity DataKd:  9nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262192(CHEMBL4083840)
Affinity DataKd:  9nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50092312(Birabresib | MK-8628 | OTX-015)
Affinity DataIC50: 16nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262195(CHEMBL4076398)
Affinity DataIC50: 17nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 61nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262192(CHEMBL4083840)
Affinity DataIC50: 68nMAssay Description:Inhibition of BRD4 BD1-BD2 (unknown origin) using tetraacetylated histone peptide as substrate after 2 hrs by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262149(CHEMBL4101842)
Affinity DataIC50: 97nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262141(CHEMBL4068474)
Affinity DataIC50: 120nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262146(CHEMBL4071890)
Affinity DataIC50: 160nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262148(CHEMBL4091132)
Affinity DataIC50: 200nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262193(CHEMBL4098881)
Affinity DataIC50: 350nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262147(CHEMBL4063264)
Affinity DataIC50: 530nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262180(CHEMBL4091003)
Affinity DataIC50: 640nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262181(CHEMBL4064879)
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262142(CHEMBL4089036)
Affinity DataIC50: 2.70E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262194(CHEMBL4073204)
Affinity DataIC50: 6.40E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262145(CHEMBL4090231)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262144(CHEMBL4079914)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262143(CHEMBL4097941)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50262196(CHEMBL4069169)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2020
Entry Details Article
PubMed