Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50001991
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451685(CHEMBL4208504)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451673(CHEMBL4202432)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451678(CHEMBL4218267)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451679(CHEMBL4214634)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451678(CHEMBL4218267)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451677(CHEMBL4204030)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451672(CHEMBL4216534)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451677(CHEMBL4204030)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451672(CHEMBL4216534)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451688(CHEMBL4213557)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451673(CHEMBL4202432)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451680(CHEMBL4207218)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451685(CHEMBL4208504)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451681(CHEMBL4208198)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451681(CHEMBL4208198)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451680(CHEMBL4207218)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451688(CHEMBL4213557)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451676(CHEMBL4214898)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451679(CHEMBL4214634)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451674(CHEMBL4208875)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451676(CHEMBL4214898)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451671(CHEMBL4205366)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451687(CHEMBL4214123)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451687(CHEMBL4214123)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451674(CHEMBL4208875)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451686(CHEMBL4211162)
Affinity DataIC50: 12nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451675(CHEMBL4218705)
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451684(CHEMBL4203994)
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451671(CHEMBL4205366)
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK6 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451682(CHEMBL4213770)
Affinity DataIC50: 36nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451677(CHEMBL4204030)
Affinity DataIC50: 36nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451678(CHEMBL4218267)
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451673(CHEMBL4202432)
Affinity DataIC50: 97nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451672(CHEMBL4216534)
Affinity DataIC50: 101nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451688(CHEMBL4213557)
Affinity DataIC50: 103nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451680(CHEMBL4207218)
Affinity DataIC50: 134nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451685(CHEMBL4208504)
Affinity DataIC50: 136nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451679(CHEMBL4214634)
Affinity DataIC50: 140nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451687(CHEMBL4214123)
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451674(CHEMBL4208875)
Affinity DataIC50: 231nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451683(CHEMBL4206797)
Affinity DataIC50: 283nMAssay Description:Inhibition of CDK4 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451681(CHEMBL4208198)
Affinity DataIC50: 301nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451676(CHEMBL4214898)
Affinity DataIC50: 412nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451671(CHEMBL4205366)
Affinity DataIC50: 801nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451684(CHEMBL4203994)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50110183(Abemaciclib | LY-2835219 | US10696678, Example LY2...)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451686(CHEMBL4211162)
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Shanghai Haihe Pharmaceutial

Curated by ChEMBL
LigandPNGBDBM50451675(CHEMBL4218705)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of CDK1 (unknown origin) using U-light as substrate preincubated for 1 hr followed by EDTA addition measured after 1 hr by LANCE Ultra kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
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