Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50035772
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020299((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-7-phenyl-h...)
Affinity DataIC50: 32nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50035622(l-Prostaglandin F2-alpha | (5Z,13E,15S)-9alpha,11a...)
Affinity DataIC50: 43nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50405735(CHEMBL2114230)
Affinity DataIC50: 71nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50035622(l-Prostaglandin F2-alpha | (5Z,13E,15S)-9alpha,11a...)
Affinity DataIC50: 140nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020299((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-7-phenyl-h...)
Affinity DataIC50: 240nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020302(CHEMBL88974 | (S-isomer)7-{2-[5-(4-Azido-phenyl)-3...)
Affinity DataIC50: 330nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020303(CHEMBL90450 | (S-isomer)7-{2-[5-(4-Azido-3-iodo-ph...)
Affinity DataIC50: 350nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50405735(CHEMBL2114230)
Affinity DataIC50: 670nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020301(CHEMBL422242 | (R-isomer)7-[3,5-Dihydroxy-2-(3-hyd...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020306(CHEMBL315519 | (S-isomer)7-{2-[5-(4-Azido-2-hydrox...)
Affinity DataIC50: 6.10E+3nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020303(CHEMBL90450 | (S-isomer)7-{2-[5-(4-Azido-3-iodo-ph...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020302(CHEMBL88974 | (S-isomer)7-{2-[5-(4-Azido-phenyl)-3...)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020305(CHEMBL89096 | (R-isomer)7-{2-[4-(3-Azido-5-hydroxy...)
Affinity DataIC50: 1.10E+4nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50405737(CHEMBL2114229)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50405736(CHEMBL2114224)
Affinity DataIC50: 6.80E+4nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020304(CHEMBL422418 | (R-isomer)7-{2-[4-(4-Azido-2-hydrox...)
Affinity DataIC50: 1.20E+5nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Bovine)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020306(CHEMBL315519 | (S-isomer)7-{2-[5-(4-Azido-2-hydrox...)
Affinity DataIC50: 2.20E+5nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed