Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50002009
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50452090(CHEMBL4218201)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50452088(CHEMBL4216755)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50452091(CHEMBL4207007)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50452087(CHEMBL4211226)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50452086(CHEMBL4218975)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50334594(2-(5-chloro-2-(2-methoxy-4-morpholinophenylamino)p...)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFocal adhesion kinase 1(Human)
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50452089(CHEMBL4209502)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FAK cytoplasmic domain (393 to 698 residues) expressed in baculovirus infected sf9 cells assess...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed