Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50002137
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020475(CHEMBL341192 | [7-Methyl-5-(thiophene-2-carbonyl)-...)
Affinity DataIC50: 860nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020464(CHEMBL135161 | [5-(2-Methoxycarbonylamino-1H-benzo...)
Affinity DataIC50: 880nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020463(CHEMBL134126 | Benzoic acid 5-(2-methoxycarbonylam...)
Affinity DataIC50: 1.95E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020478(CHEMBL133799 | [5-(4-Cyanomethyl-thiophene-2-carbo...)
Affinity DataIC50: 2.90E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020459(CHEMBL336862 | [5-(2-Methoxycarbonylamino-1H-benzo...)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020480(CHEMBL422615 | [5-(2-Methoxycarbonylamino-1H-benzo...)
Affinity DataIC50: 5.20E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM97233(cid_4122 | MLS001164242 | SMR000326904 | Nocodazol...)
Affinity DataIC50: 5.70E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020479(CHEMBL133900 | [5-(2-Methoxycarbonylamino-1H-benzo...)
Affinity DataIC50: 7.50E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020460(CHEMBL132946 | 2,2,2-Trifluoro-1-[5-(2-methoxycarb...)
Affinity DataIC50: 8.30E+3nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020461(CHEMBL422269 | [5-(Thiophene-2-carbonyl)-1H-benzoi...)
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020469(CHEMBL134616 | {5-[4-(2,2,2-Trifluoro-acetyl)-thio...)
Affinity DataIC50: 1.60E+4nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020474(CHEMBL133155 | [5-(4-Methyl-thiophene-2-carbonyl)-...)
Affinity DataIC50: 1.76E+4nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020455(CHEMBL130090 | [5-(4-Hydroxymethyl-thiophene-2-car...)
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020454(CHEMBL133877 | {5-[4-(tert-Butoxycarbonylamino-met...)
Affinity DataIC50: 2.33E+4nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020473(CHEMBL135796 | [4-Methyl-5-(thiophene-2-carbonyl)-...)
Affinity DataIC50: 1.06E+5nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020472(CHEMBL336324 | [5-(4-Aminomethyl-thiophene-2-carbo...)
Affinity DataIC50: 1.20E+5nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTubulin alpha-1A chain(Pig)
Smith Kline & French Laboratories

Curated by ChEMBL
LigandPNGBDBM50020468(CHEMBL130169 | [5-(2-Methoxycarbonylamino-1H-benzo...)
Affinity DataIC50: 4.42E+5nMAssay Description:Displacement of 5.8 uM [3H]-oncodazole from homogeneous tubulin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed