Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50002892
TargetP2X purinoceptor 7(Human)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464474(CHEMBL4281588)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464474(CHEMBL4281588)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464477(CHEMBL4292211)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464477(CHEMBL4292211)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50234965(A-740003 | N-(1-{[(Cyanoimino)(5-quinolinylamino)m...)
Affinity DataIC50: 109nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464475(CHEMBL4291798)
Affinity DataIC50: 414nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50277548(CHEMBL4173394)
Affinity DataIC50: 536nMAssay Description:Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464475(CHEMBL4291798)
Affinity DataIC50: 712nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50234965(A-740003 | N-(1-{[(Cyanoimino)(5-quinolinylamino)m...)
Affinity DataIC50: 897nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464471(CHEMBL4293271)
Affinity DataIC50: 3.17E+3nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50277548(CHEMBL4173394)
Affinity DataIC50: 1.52E+4nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464472(CHEMBL4285010)
Affinity DataIC50: 3.35E+4nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464470(CHEMBL4290432)
Affinity DataIC50: 4.58E+4nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50049066(CHEBI:44401 | 2-Hydroxynaphthoquinone | Lawsone | ...)
Affinity DataIC50: 7.55E+4nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464476(CHEMBL4285438)
Affinity DataIC50: 8.01E+4nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Mouse)
Instituto Oswaldo Cruz

Curated by ChEMBL
LigandPNGBDBM50464473(CHEMBL1341602)
Affinity DataIC50: 8.13E+4nMAssay Description:Antagonist activity at P2X7R in Swiss Webster mouse peritoneal macrophages assessed as inhibition of ATP-induced propidium iodide uptake preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed