Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50018704
TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb Research and Development
Curated by ChEMBL
Bristol-Myers Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 8.5nMAssay Description:Inhibition of human Nav 1.7 channel expressed in HEK293 cells at -10 mV holding potential by whole cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb Research and Development
Curated by ChEMBL
Bristol-Myers Squibb Research and Development
Curated by ChEMBL
Affinity DataIC50: 907nMAssay Description:Inhibition of human Nav 1.7 channel expressed in HEK293 cells at -10 mV holding potential by whole cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity to human V1a assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human V1a assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to human V1a assessed as inhibition constantMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Human)
Bristol-Myers Squibb Research and Development
Curated by ChEMBL
Bristol-Myers Squibb Research and Development
Curated by ChEMBL
Affinity DataKi: 273nMAssay Description:Binding affinity to human recombinant ALK L1196M mutant (1093 to 1411 residues) assessed as inhibition constant using 5'FAM-KKSRGDYMTMQIG-CONH2 pepti...More data for this Ligand-Target Pair
