Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50002154
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50121933(Ac-Phe-Phe-Phe-Arg-Leu-Arg-Arg-D-Ala-Arg-Pro-Lys-N...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454178(CHEMBL4214138)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454176(CHEMBL4217438)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454179(CHEMBL4217592)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454181(CHEMBL4206658)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454177(CHEMBL4204599)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454180(CHEMBL4202742)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454178(CHEMBL4214138)
Affinity DataKi:  903nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454181(CHEMBL4206658)
Affinity DataKi:  1.17E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454177(CHEMBL4204599)
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454176(CHEMBL4217438)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50121933(Ac-Phe-Phe-Phe-Arg-Leu-Arg-Arg-D-Ala-Arg-Pro-Lys-N...)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454179(CHEMBL4217592)
Affinity DataKi:  1.92E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50454180(CHEMBL4202742)
Affinity DataKi:  3.46E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Kansas

Curated by ChEMBL
LigandPNGBDBM50121933(Ac-Phe-Phe-Phe-Arg-Leu-Arg-Arg-D-Ala-Arg-Pro-Lys-N...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]DPDPE from rat delta opioid receptor expressed in CHO cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed