Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50002165
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Jilin University

Curated by ChEMBL
LigandPNGBDBM349364((4R)-6-(1-tert-butylpyrazol-4- | US10206931, Examp...)
Affinity DataIC50: 470nMAssay Description:Inhibition of human His-FLAG tagged CBP/EP300 (1082 to 1197 residues) using H4-TetraAc-biotin peptide as substrate after 90 mins by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Jilin University

Curated by ChEMBL
LigandPNGBDBM50178216(CHEMBL3814920 | US10206931, Example 131)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human His-FLAG tagged CBP/EP300 (1082 to 1197 residues) using H4-TetraAc-biotin peptide as substrate after 90 mins by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed