Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50001672
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292270(CHEMBL4163588)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50387881(CHEMBL2057799)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292266(CHEMBL4169388)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataIC50: 120nMAssay Description:Neutral antagonist activity at human CB2 assessed as restoration of forskolin-induced cAMP formation preincubated for 15 mins followed by forskolin a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataIC50: 120nMAssay Description:Neutral antagonist activity at human CB2 assessed as inhibition of WIN552122-induced suppression of cAMP formation preincubated for 15 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292265(CHEMBL4177237)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292267(CHEMBL4162105)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292278(CHEMBL4174271)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292279(CHEMBL4176159)
Affinity DataKi:  329nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292269(CHEMBL4165549)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292280(CHEMBL4168970)
Affinity DataKi:  678nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292270(CHEMBL4163588)
Affinity DataIC50: 930nMAssay Description:Neutral antagonist activity at human CB2 assessed as inhibition of WIN552122-induced suppression of cAMP formation preincubated for 15 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292270(CHEMBL4163588)
Affinity DataIC50: 930nMAssay Description:Neutral antagonist activity at human CB2 assessed as restoration of forskolin-induced cAMP formation preincubated for 15 mins followed by forskolin a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292264(CHEMBL4172723)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292281(CHEMBL4161047)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292258(CHEMBL4164392)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292259(CHEMBL4166726)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292256(CHEMBL4167826)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292257(CHEMBL4175043)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292262(CHEMBL4171188)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292263(CHEMBL4164823)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292260(CHEMBL4174629)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292261(CHEMBL4163287)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292265(CHEMBL4177237)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292266(CHEMBL4169388)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292263(CHEMBL4164823)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292264(CHEMBL4172723)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292269(CHEMBL4165549)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292267(CHEMBL4162105)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292268(CHEMBL4172780)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292257(CHEMBL4175043)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292258(CHEMBL4164392)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292268(CHEMBL4172780)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292256(CHEMBL4167826)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292261(CHEMBL4163287)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292262(CHEMBL4171188)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292259(CHEMBL4166726)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292260(CHEMBL4174629)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292280(CHEMBL4168970)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292281(CHEMBL4161047)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292279(CHEMBL4176159)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50387881(CHEMBL2057799)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50160434(AM630 | (6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50292270(CHEMBL4163588)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-CP-55940 from human CB1 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2020
Entry Details Article
PubMed