Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50002181
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454721(CHEMBL4217182)
Affinity DataEC50:  0.700nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454706(CHEMBL4214528)
Affinity DataEC50:  0.900nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454714(CHEMBL4209188)
Affinity DataEC50:  1.20nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454708(CHEMBL4213342)
Affinity DataEC50:  2.20nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454723(CHEMBL4202871)
Affinity DataEC50:  6.20nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataIC50: 7nMAssay Description:Antagonistic activity at 5-HT2c receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454721(CHEMBL4217182)
Affinity DataIC50: 8nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454719(CHEMBL4210030)
Affinity DataEC50:  9nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454710(CHEMBL4205772)
Affinity DataIC50: 9.30nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataIC50: 10nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454708(CHEMBL4213342)
Affinity DataIC50: 11nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454719(CHEMBL4210030)
Affinity DataIC50: 11nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454717(CHEMBL4214642)
Affinity DataIC50: 11nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454718(CHEMBL4202443)
Affinity DataEC50:  11nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454717(CHEMBL4214642)
Affinity DataEC50:  13nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454707(CHEMBL4217986)
Affinity DataEC50:  17nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454722(CHEMBL4210637)
Affinity DataEC50:  18nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454714(CHEMBL4209188)
Affinity DataIC50: 24nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataEC50:  24nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454702(CHEMBL4207328)
Affinity DataEC50:  24nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454706(CHEMBL4214528)
Affinity DataIC50: 27nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454720(CHEMBL4212622)
Affinity DataEC50:  28nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataIC50: 32nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454722(CHEMBL4210637)
Affinity DataIC50: 38nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454717(CHEMBL4214642)
Affinity DataIC50: 42nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454713(CHEMBL4205326)
Affinity DataEC50:  42nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454707(CHEMBL4217986)
Affinity DataIC50: 43nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454703(CHEMBL4217039)
Affinity DataIC50: 43nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454702(CHEMBL4207328)
Affinity DataIC50: 51nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454716(CHEMBL4215048)
Affinity DataIC50: 52nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454711(CHEMBL4210128)
Affinity DataIC50: 52nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454711(CHEMBL4210128)
Affinity DataIC50: 54nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454720(CHEMBL4212622)
Affinity DataIC50: 54nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454704(CHEMBL4218526)
Affinity DataIC50: 59nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454719(CHEMBL4210030)
Affinity DataIC50: 60nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454712(CHEMBL4204832)
Affinity DataIC50: 62nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454719(CHEMBL4210030)
Affinity DataIC50: 63nMAssay Description:Antagonistic activity at 5-HT2c receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454721(CHEMBL4217182)
Affinity DataIC50: 65nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454723(CHEMBL4202871)
Affinity DataIC50: 65nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454715(CHEMBL4209705)
Affinity DataIC50: 66nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454715(CHEMBL4209705)
Affinity DataIC50: 68nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454708(CHEMBL4213342)
Affinity DataIC50: 70nMAssay Description:Antagonistic activity at 5-HT2c receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454708(CHEMBL4213342)
Affinity DataIC50: 71nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454705(CHEMBL4213586)
Affinity DataIC50: 83nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454713(CHEMBL4205326)
Affinity DataIC50: 85nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454718(CHEMBL4202443)
Affinity DataIC50: 86nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454716(CHEMBL4215048)
Affinity DataIC50: 89nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Lance Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454703(CHEMBL4217039)
Affinity DataIC50: 90nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454704(CHEMBL4218526)
Affinity DataIC50: 94nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50454722(CHEMBL4210637)
Affinity DataIC50: 96nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
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