Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50000273
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50244503(CHEMBL4078293)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells by automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2019
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
University of Auckland

Curated by ChEMBL
LigandPNGBDBM50244503(CHEMBL4078293)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes assessed as decrease in formation of 6beta-hydroxytestosterone from testosterone after 10 mins by LC-M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2019
Entry Details Article
PubMed