Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50002592
TargetNuclear receptor ROR-gamma(Human)
University of Padova

Curated by ChEMBL
LigandPNGBDBM50460230(CHEMBL4225360)
Affinity DataIC50: 4.40E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) expressed in HEK293 cells measured after 48 hrs post transfection by dual-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
University of Padova

Curated by ChEMBL
LigandPNGBDBM50460229(CHEMBL4229166)
Affinity DataIC50: 4.70E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) expressed in HEK293 cells measured after 48 hrs post transfection by dual-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
University of Padova

Curated by ChEMBL
LigandPNGBDBM50460232(CHEMBL4226196)
Affinity DataIC50: 6.50E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) expressed in HEK293 cells measured after 48 hrs post transfection by dual-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
University of Padova

Curated by ChEMBL
LigandPNGBDBM50460231(CHEMBL4225089)
Affinity DataIC50: 6.80E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORgammat LBD (unknown origin) expressed in HEK293 cells measured after 48 hrs post transfection by dual-lucif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed