Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50002425
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458422(CHEMBL4216958)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458415(CHEMBL567508 | EN300-02284)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458419(CHEMBL4203286)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458417(CHEMBL4203489)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458416(CHEMBL1230155)
Affinity DataKd:  9.00E+5nMAssay Description:Binding affinity to 15N-Gly/Cys/Ser/Trp-labeled human USP2a expressed in Escherichia coli BL21(DE3) assessed as change in chemical shift by NMR metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458416(CHEMBL1230155)
Affinity DataIC50: 1.30E+6nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458421(CHEMBL1650269)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458420(CHEMBL4207620)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 2(Human)
Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50458418(CHEMBL4207578)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of human USP2a (258 to 605 residues) expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate incubated for 30 mins measured at 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed