Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002970
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM24567(Tetrahydrolipstatin | CHEMBL175247 | Xenical | (2S...)
Affinity DataIC50: 4nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465318(CHEMBL472695)
Affinity DataIC50: 8nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465320(CHEMBL4282840)
Affinity DataIC50: 15nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465321(CHEMBL4291122)
Affinity DataIC50: 15nMAssay Description:Inhibition of porcine pancreatic lipaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50274723(N-Formyl-D-leucine-(1S)-1-[[(2S,3S)-3-hexyl-4-oxo-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465317(CHEMBL4282614)
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465323(CHEMBL4282318)
Affinity DataIC50: 20nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465319(CHEMBL4290524)
Affinity DataIC50: 77nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM24567(Tetrahydrolipstatin | CHEMBL175247 | Xenical | (2S...)
Affinity DataIC50: 360nMAssay Description:Inhibition of porcine pancreatic lipase using triolein as substrate measured after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPancreatic triacylglycerol lipase(Pig)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50465322(CHEMBL2305145)
Affinity DataIC50: 930nMAssay Description:Inhibition of porcine pancreatic lipase using p-nitrophenyl butyrate as substrate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed