Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50002631
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460764(CHEMBL77772)
Affinity DataEC50:  60nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460764(CHEMBL77772)
Affinity DataEC50:  60nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  870nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  871nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460760(CHEMBL4228433)
Affinity DataEC50:  3.69E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460760(CHEMBL4228433)
Affinity DataEC50:  3.72E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460761(CHEMBL4227443)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460761(CHEMBL4227443)
Affinity DataEC50:  4.93E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460759(CHEMBL4226014)
Affinity DataEC50:  5.89E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460759(CHEMBL4226014)
Affinity DataEC50:  5.93E+3nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460763(CHEMBL4228169)
Affinity DataEC50:  1.86E+4nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460763(CHEMBL4228169)
Affinity DataEC50:  1.87E+4nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50136847(Octanoic acid [2-(4-hydroxy-phenyl)-ethyl]-amide |...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50136847(Octanoic acid [2-(4-hydroxy-phenyl)-ethyl]-amide |...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460762(CHEMBL4226595)
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Mannheim University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50460762(CHEMBL4226595)
Affinity DataEC50: >5.01E+5nMAssay Description:Agonist activity at recombinant TRPV1 (unknown origin) expressed in HEK293 cells assessed as induction of calcium flux administered for 1 min followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed