Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50002656
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | Chlorochin | CHLOROQUINE PHOSPHATE | Chlo...)
Affinity DataIC50: 20nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | Chlorochin | CHLOROQUINE PHOSPHATE | Chlo...)
Affinity DataIC50: 200nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461234(CHEMBL4226443)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461235(CHEMBL4227918)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461235(CHEMBL4227918)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461234(CHEMBL4226443)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461226(CHEMBL4228534)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461226(CHEMBL4228534)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461225(CHEMBL4224867)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461237(CHEMBL4226863)
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461229(CHEMBL4228490)
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461239(CHEMBL4227712)
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461233(CHEMBL4224976)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461237(CHEMBL4226863)
Affinity DataIC50: 2.53E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461236(CHEMBL4228011)
Affinity DataIC50: 2.67E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461225(CHEMBL4224867)
Affinity DataIC50: 2.67E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461232(CHEMBL4227123)
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461229(CHEMBL4228490)
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461236(CHEMBL4228011)
Affinity DataIC50: 2.99E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461239(CHEMBL4227712)
Affinity DataIC50: 3.04E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461232(CHEMBL4227123)
Affinity DataIC50: 3.38E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461230(CHEMBL4224721)
Affinity DataIC50: 3.42E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461233(CHEMBL4224976)
Affinity DataIC50: 4.16E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461230(CHEMBL4224721)
Affinity DataIC50: 4.45E+4nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461227(CHEMBL4228230)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461228(CHEMBL4226325)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461228(CHEMBL4226325)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461238(CHEMBL4224700)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461227(CHEMBL4228230)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain-2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461231(CHEMBL4228548)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine resistant Plasmodium falciparum RKL9 schizont stage infected in human erythrocytes assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461238(CHEMBL4224700)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Delhi Institute of Pharmaceutical Sciences and Research

Curated by ChEMBL
LigandPNGBDBM50461231(CHEMBL4228548)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of falcipain-2 in chloroquine sensitive Plasmodium falciparum MRC-02 schizont stage infected in human erythrocytes assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed