Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50002673
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461446(CHEMBL4227742)
Affinity DataIC50: 230nMAssay Description:Inhibition of African green monkey SOAT1 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461446(CHEMBL4227742)
Affinity DataIC50: 780nMAssay Description:Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461446(CHEMBL4227742)
Affinity DataIC50: 860nMAssay Description:Inhibition of African green monkey SOAT2 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461447(CHEMBL4228016)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of African green monkey SOAT1 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50360305(CHEMBL409855 | US9149492, Beauveriolide III)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461447(CHEMBL4228016)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461448(CHEMBL4227559)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of African green monkey SOAT1 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461447(CHEMBL4228016)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461446(CHEMBL4227742)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50360305(CHEMBL409855 | US9149492, Beauveriolide III)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of African green monkey SOAT1 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50360305(CHEMBL409855 | US9149492, Beauveriolide III)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of African green monkey SOAT2 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461447(CHEMBL4228016)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of African green monkey SOAT2 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461448(CHEMBL4227559)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461448(CHEMBL4227559)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of African green monkey SOAT1 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50461448(CHEMBL4227559)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of African green monkey SOAT2 isolated from CHO cell microsomes assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 5 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Green monkey)
Tohoku Medical and Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50360305(CHEMBL409855 | US9149492, Beauveriolide III)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of African green monkey SOAT2 expressed in CHO cells assessed as decrease in [14C]CE synthesis from [14C]oleic acid after 6 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed