Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002682
TargetGlucose-dependent insulinotropic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461586(CHEMBL4229220)
Affinity DataEC50:  25nMAssay Description:Agonist activity at GPR119 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461585(CHEMBL4224878)
Affinity DataEC50:  2nMAssay Description:Agonist activity at GPR119 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461582(CHEMBL4225726)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GPR119 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461581(CHEMBL3133098)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of DGAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461587(CHEMBL3133093)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of DGAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461583(CHEMBL3133094)
Affinity DataIC50: 100nMAssay Description:Inhibition of DGAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50461584(CHEMBL3133100)
Affinity DataIC50: 631nMAssay Description:Inhibition of DGAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50461582(CHEMBL4225726)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50461585(CHEMBL4224878)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50461586(CHEMBL4229220)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed