Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50001823
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM328993(US9663503, Compound 1 | 5-[[4-[[(2R)-morpholin-2-y...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50389803(CHEMBL2041933 | AZD7762)
Affinity DataIC50: 6nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50393330(CHEMBL4175978)
Affinity DataIC50: 684nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50379285(CHEMBL4164408)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50379262(CHEMBL4170449)
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50389840(CHEMBL4176499)
Affinity DataIC50: 2.83E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50391340(CHEMBL4176473)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50379263(CHEMBL4177166)
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50394673(CHEMBL4174578)
Affinity DataIC50: 8.06E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50398335(CHEMBL4166347)
Affinity DataIC50: 9.87E+3nMAssay Description:Inhibition of CHK1 (unknown origin) using Cdc25 peptide as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed