Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 4777
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM30130(Prozac | cid_62857 | Fluoxetin | CHEMBL41 | CHEMBL...)
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM82217([4-(3,4-Dichloro-phenyl)-1,2,3,4-tetrahydro-naphth...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50020707(CHEMBL287064 | Nomelidine | [3-(4-Bromo-phenyl)-3-...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  9.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM66978(Zimelidine (E-isomer) | Zimelidine (Z-isomer) | (E...)
Affinity DataKi:  77.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM35229(Desmethylimipramine | 3-(10,11-dihydro-5H-dibenzo[...)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM66978(Zimelidine (E-isomer) | Zimelidine (Z-isomer) | (E...)
Affinity DataKi:  2.28E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50031942(CHEMBL1065 | Sansert | (6aR,9R)-4-Methyl-4,6,6a,7,...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Veterans Administration Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed