Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50001284
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human CDK9/CyclinT using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 300nMAssay Description:Inhibition of human PKCbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human CDK2/Cyclin A using ATP and Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of recombinant human PIM1 using CREBtide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human Aurora-B using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of mouse CLK1 using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of recombinant human PIM1 using CREBtide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of rat Dyrk1a using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human haspin using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1epsilon using Ulight-ARTKQTARKSTGGKAPRKQLAGCG as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Aurora-B using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Aurora-B using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human PIM1 using CREBtide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human haspin using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse CLK1 using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat Dyrk1a using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat Dyrk1a using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
Target[Tau protein] kinase(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3alpha using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
Target[Tau protein] kinase(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3alpha using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3beta using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3beta using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3beta using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1epsilon using Ulight-ARTKQTARKSTGGKAPRKQLAGCG as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse CLK1 using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1epsilon using Ulight-ARTKQTARKSTGGKAPRKQLAGCG as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human haspin using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
Target[Tau protein] kinase(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3alpha using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1epsilon using Ulight-ARTKQTARKSTGGKAPRKQLAGCG as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Aurora-B using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human PIM1 using CREBtide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human haspin using full-length histone H3 as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse CLK1 using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat Dyrk1a using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3beta using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase 1, delta tv1(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50256734((-)-Cercosporamide | CHEMBL475816)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase 1, delta tv1(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK2/Cyclin A using ATP and Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
Target[Tau protein] kinase(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig GSK3alpha using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 60 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase 1, delta tv1(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK2/Cyclin A using ATP and Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274761(CHEMBL4127885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK2/Cyclin A using ATP and Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 30 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCasein kinase 1, delta tv1(Pig)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274742(CHEMBL4129279)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of pig CK1deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50274762(CHEMBL4128587)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human CDK9/CyclinT using Ulight-CFFKNIVTPRTPPPSQGK-amide as substrate after 90 mins by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2020
Entry Details Article
PubMed