Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50001291
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataKi:  0.269nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataKi:  0.871nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275109(CHEMBL4128853)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275109(CHEMBL4128853)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275109(CHEMBL4128853)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275109(CHEMBL4128853)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity to DOR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275109(CHEMBL4128853)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275109(CHEMBL4128853)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275110(CHEMBL4130069)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275110(CHEMBL4130069)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]DAMGO from MOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataEC50:  11.7nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)
Affinity DataKi:  12nMAssay Description:Binding affinity to MOR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataEC50:  12nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataEC50:  13nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275107(CHEMBL4130303)
Affinity DataEC50:  14nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275110(CHEMBL4130069)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275110(CHEMBL4130069)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]U69593 from KOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275110(CHEMBL4130069)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275110(CHEMBL4130069)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DADLE from DOR (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataEC50:  27nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataEC50:  27nMAssay Description:Agonist activity at DOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataEC50:  63nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataEC50:  63nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataEC50:  87nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataEC50:  87nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataEC50:  112nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275111(CHEMBL4126803)
Affinity DataEC50:  112nMAssay Description:Agonist activity at MOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataEC50:  135nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50275108(CHEMBL4129668)
Affinity DataEC50:  135nMAssay Description:Agonist activity at KOR (unknown origin) expressed in HEK cells assessed as reduction in cAMP accumulation by split luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2020
Entry Details Article
PubMed
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