Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50018712
Affinity DataIC50: 0.100nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of LIMK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit gamma(Human)
Universita Degli Studi Di Siena
Curated by ChEMBL
Universita Degli Studi Di Siena
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of ROCK2 (unknown origin) by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 200 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 25 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of CHK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human LIMK1 (312 to 638 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human LIMK1 (312 to 638 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human LIMK1 (312 to 638 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of LIMK1 (unknown origin) phosphorylation of cofilinMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Inhibition of ROCK2 (unknown origin) by Kinase Glo luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human LIMK1 (312 to 638 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant ROCK2 by ADP glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant LIMK1 in presence of ATP cofilin as substrate at 25 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of LIMK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of LIMK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of LIMK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant LIMK1 in presence of ATP cofilin as substrate at 25 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant LIMK1 in presence of ATP cofilin as substrate at 25 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant LIMK1 in presence of ATP cofilin as substrate at 25 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of human LIMK1 (312 to 638 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of LIMK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant LIMK1More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant LIMK1 in presence of ATP cofilin as substrate at 25 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant ROCK2 by ADP glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of human recombinant LIMK2More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of human LIMK1 (321 to 647 residues) expressed in Sf9 cells using dextrin as substrate incubated for 30 mins by micro-scintillation fluid ...More data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Inhibition of human recombinant LIMK2More data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Inhibition of LIMK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of LIMK2 (unknown origin) in presence of ATP at 25 uMMore data for this Ligand-Target Pair
































