Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50003255
TargetKinesin-like protein KIF11(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50216514(4-(3-hydroxyphenyl)-7,7-dimethyl-2-thioxo-1,2,3,4,...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Eg5More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human VEGFR-2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase mTOR(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataIC50: 430nMAssay Description:Inhibition of mTOR (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50468599(CHEMBL4291192)
Affinity DataIC50: 640nMAssay Description:Inhibition of mTOR (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50468598(CHEMBL4286023)
Affinity DataIC50: 720nMAssay Description:Inhibition of mTOR (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50468598(CHEMBL4286023)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human VEGFR-2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50468599(CHEMBL4291192)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of human VEGFR-2 incubated for 2.5 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetKinesin-like protein KIF11(Human)
Mansoura University

Curated by ChEMBL
LigandPNGBDBM50468600(CHEMBL444096)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human Eg5More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed