Report error Found 121 Enz. Inhib. hit(s) with all data for entry = 50002465
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Antagonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 93nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Binding affinity to human ERbeta LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Binding affinity to human ERalpha LBD after 2 hrs in absence of light by competitive fluorometric binding assayMore data for this Ligand-Target Pair
