Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50002808
TargetLarge neutral amino acids transporter small subunit 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50463321(CHEMBL4239455)
Affinity DataIC50: 2.77E+4nMAssay Description:Inhibition of LAT1-mediated [14C]-L-leucine uptake in human MCF7 cells after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLarge neutral amino acids transporter small subunit 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50463322(CHEMBL4242544)
Affinity DataIC50: 3.24E+4nMAssay Description:Inhibition of LAT1-mediated [14C]-L-leucine uptake in human MCF7 cells after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetLarge neutral amino acids transporter small subunit 1(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM60928(L-DOPA | dihydroxyphenylalanine | BDBM50130192 | L...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of LAT1-mediated [14C]-L-leucine uptake in human MCF7 cells after 5 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)