Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50003104
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467028(CHEMBL4281089)
Affinity DataIC50: 900nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467029(CHEMBL4285364)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467033(CHEMBL4279547)
Affinity DataIC50: 6.90E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467030(CHEMBL4290212)
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467031(CHEMBL4276988)
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Janssen Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50467032(CHEMBL4284935)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of 3H-dofetilide from human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed