Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50003115
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467129(CHEMBL4278280)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467130(CHEMBL4291216)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467140(CHEMBL4289788)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467133(CHEMBL4280574)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467135(CHEMBL4287379)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467138(CHEMBL4282931)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364573(CHEMBL1951143)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467139(CHEMBL4293170)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467136(CHEMBL4284022)
Affinity DataIC50: 5.60nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467134(CHEMBL4284403)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467137(CHEMBL4294618)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467132(CHEMBL4292297)
Affinity DataIC50: 70nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed