Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50001931
TargetShort transient receptor potential channel 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50450630(CHEMBL101896)
Affinity DataIC50: 300nMAssay Description:Modulation of TRPC1/TRPC3/STIM1/Orai1 in HEK cells assessed as induction of store-operated calcium entry by measuring residual activity preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetShort transient receptor potential channel 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50450629(CHEMBL4177187)
Affinity DataIC50: 500nMAssay Description:Modulation of TRPC1/TRPC3/STIM1/Orai1 in HEK cells assessed as induction of store-operated calcium entry by measuring residual activity preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
LigandPNGBDBM50450626(CHEMBL4162723)
Affinity DataIC50: 600nMAssay Description:Modulation of TRPC1/TRPC3/STIM1/Orai1 in HEK cells assessed as induction of store-operated calcium entry by measuring residual activity preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetStromal interaction molecule 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50450629(CHEMBL4177187)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of STIM1/STIM2/Orai1 (unknown origin) expressed in mouse BV2 cells assessed as reduction of store-operated calcium entry at 100 uM preincu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetShort transient receptor potential channel 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50450627(CHEMBL4162062)
Affinity DataIC50: 3.10E+3nMAssay Description:Modulation of TRPC1/TRPC3/STIM1/Orai1 in HEK cells assessed as induction of store-operated calcium entry by measuring residual activity preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetShort transient receptor potential channel 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50450628(CHEMBL4172741)
Affinity DataIC50: 4.40E+3nMAssay Description:Modulation of TRPC1/TRPC3/STIM1/Orai1 in HEK cells assessed as induction of store-operated calcium entry by measuring residual activity preincubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetStromal interaction molecule 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50450626(CHEMBL4162723)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of STIM1/STIM2/Orai1 (unknown origin) expressed in mouse BV2 cells assessed as induction of store-operated calcium entry by measuring resi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed