Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50003068
TargetSialidase(Vibrio cholerae serotype O1 (strain ATCC 39315 / E...)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Vibrio cholerae serotype O1 (strain ATCC 39315 / E...)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Vibrio cholerae serotype O1 (strain ATCC 39315 / E...)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase-2(Human)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Vibrio cholerae serotype O1 (strain ATCC 39315 / E...)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Vibrio cholerae serotype O1 (strain ATCC 39315 / E...)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50: 2.89E+4nMAssay Description:Inhibition of Vibrio cholerae sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50: 4.43E+4nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase-2(Human)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase-2(Human)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase(Clostridium perfringens)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Clostridium perfringens sialidase using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase A(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Streptococcus pneumoniae NanA using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase B(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae sialidase NanC using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase B(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae sialidase NanC using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase B(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae sialidase NanC using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase-2(Human)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase NanB(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae NanB using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase B(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466473(CHEMBL4278803)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae sialidase NanC using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase B(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae sialidase NanC using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase NanB(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466472(CHEMBL4289476)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae NanB using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase NanB(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50331692((2R,3R,4S)-3-acetamido-2-((1R,2R)-3-azido-1,2-dihy...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae NanB using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSialidase-2(Human)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant human cytosolic sialidase NEU2 using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase NanB(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM4706(2,3-didehydro-2-deoxy-N-acetylneuraminic acid | (2...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae NanB using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuraminidase NanB(Streptococcus pneumoniae)
University of California-Davis

Curated by ChEMBL
LigandPNGBDBM50466474(CHEMBL4282280)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of Streptococcus pneumoniae NanB using Neu5Acalpha2-3GalbetapNP as substrate after 30 mins by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed