Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50006840
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50304738(2-(3-((S)-1-carboxy-3-methylbutyl)ureido)pentanedi...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503760(CHEMBL4442450)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503756(CHEMBL4473741)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503754(CHEMBL4458733)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503757(CHEMBL4541841)
Affinity DataIC50: 17nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503758(CHEMBL4587808)
Affinity DataIC50: 531nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503755(CHEMBL4462654)
Affinity DataIC50: 630nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Institute of Biotechnology of The Czech Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50503759(CHEMBL4513258)
Affinity DataIC50: 8.53E+3nMAssay Description:Inhibition of N-terminally tagged human recombinant GCP2 (44 to 750 residues) extracellular domain expressed in Drosophila melanogaster S2 cells prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed