Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50006843
TargetCholinesterase(Horse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50344826(1-(4-chlorobenzyl)-3-hydroxy-3-phenylindolin-2-one...)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of AChE in Swiss mouse brain homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Horse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503820(CHEMBL4550082)
Affinity DataIC50: 6.61E+3nMAssay Description:Inhibition of equine serum BuChE after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503818(CHEMBL4593576)
Affinity DataIC50: 7.41E+3nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of equine serum BuChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCholinesterase(Horse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataKi:  4.10E+4nMAssay Description:Reversible competitive inhibition of equine BuChE by Lineweaver-burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.25E+5nMAssay Description:Inhibition of AChE in Swiss mouse liver homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Electric eel)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50344826(1-(4-chlorobenzyl)-3-hydroxy-3-phenylindolin-2-one...)
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCholinesterase(Mouse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.47E+5nMAssay Description:Inhibition of BuChE in Swiss mouse liver homogenate by Ellman's assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503820(CHEMBL4550082)
Affinity DataIC50: 1.93E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503818(CHEMBL4593576)
Affinity DataIC50: 2.37E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetCholinesterase(Mouse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50: 4.35E+5nMAssay Description:Inhibition of BuChE in Swiss mouse liver homogenate by Ellman's assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of electrophorus electricus AChEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Universidade De £Vora

Curated by ChEMBL
LigandPNGBDBM50503819(CHEMBL4565335)
Affinity DataIC50: 5.65E+5nMAssay Description:Inhibition of AChE in Swiss mouse liver homogenate using acetylthiocholine iodide as substrate by Ellman's assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed