Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50008382
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518649(CHEMBL4450967)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518649(CHEMBL4450967)
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518652(CHEMBL4539295)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518652(CHEMBL4539295)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518655(CHEMBL4457029)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518655(CHEMBL4457029)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518655(CHEMBL4457029)
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518651(CHEMBL4464233)
Affinity DataIC50: 4.26E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM71542(Primaquine bisphosphate | N4-(6-methoxy-8-quinolin...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518658(CHEMBL4476130)
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518650(CHEMBL4526451)
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518660(CHEMBL4454754)
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518659(CHEMBL4593962)
Affinity DataIC50: 2.27E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518650(CHEMBL4526451)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518654(Quinoxaline-2-Carboxylic Acid | CHEMBL151797)
Affinity DataIC50: 3.20E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518657(Quinoline-3-Carboxylic Acid | CHEMBL275098)
Affinity DataIC50: 2.40E+6nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM54704(UNM-0000306098 | cid_23681059 | sodium;(2S)-2-(6-m...)
Affinity DataIC50: 6.70E+6nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518656(CHEMBL4435617)
Affinity DataIC50: 9.60E+6nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518653(CHEBI:16533 | Trp-NH2 | CHEMBL227123)
Affinity DataIC50: 9.90E+6nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
University of Missouri-Kansas City

Curated by ChEMBL
LigandPNGBDBM50518653(CHEBI:16533 | Trp-NH2 | CHEMBL227123)
Affinity DataIC50: 1.57E+7nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as reduction in [3H]dTTP incorporation using poly(rA)/oligo(dT) as template/primer after 30 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed