Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50008389
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518734(CHEMBL4467081)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition and measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518732(CHEMBL4473488)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition and measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518733(CHEMBL4448808)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition and measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518735(CHEMBL4584218)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition and measured f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518736(CHEMBL4526940)
Affinity DataKi:  625nMAssay Description:Inhibition of recombinant Pin1 (unknown origin) using Suc-AEPF-MCA as substrate preincubated followed by substrate addition and measured after 60 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518734(CHEMBL4467081)
Affinity DataKi:  1.37E+3nMAssay Description:Irreversible inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Nagoya Citi University

Curated by ChEMBL
LigandPNGBDBM50518732(CHEMBL4473488)
Affinity DataKi:  5.47E+3nMAssay Description:Irreversible inhibition of Pin1 (unknown origin) using suc-Ala-Glu-Pro-Phe-pNA as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed