Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50008390
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518750(CHEMBL4566454)
Affinity DataEC50:  68nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518749(CHEMBL4461852)
Affinity DataEC50:  68nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518759(CHEMBL275850)
Affinity DataEC50:  77nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518759(CHEMBL275850)
Affinity DataEC50:  85nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518749(CHEMBL4461852)
Affinity DataEC50:  108nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518755(CHEMBL4450542)
Affinity DataEC50:  109nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518744(CHEMBL4591840)
Affinity DataEC50:  113nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518755(CHEMBL4450542)
Affinity DataEC50:  115nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518739(CHEMBL280106)
Affinity DataEC50:  142nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518750(CHEMBL4566454)
Affinity DataEC50:  164nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518754(CHEMBL4458039)
Affinity DataEC50:  228nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518744(CHEMBL4591840)
Affinity DataEC50:  231nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518741(CHEMBL4475354)
Affinity DataEC50:  232nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518751(CHEMBL4525895)
Affinity DataEC50:  245nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518742(CHEMBL4527494)
Affinity DataEC50:  259nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518751(CHEMBL4525895)
Affinity DataEC50:  309nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518754(CHEMBL4458039)
Affinity DataEC50:  351nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518752(CHEMBL4450521)
Affinity DataEC50:  390nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518741(CHEMBL4475354)
Affinity DataEC50:  396nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518752(CHEMBL4450521)
Affinity DataEC50:  493nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518756(CHEMBL1546037)
Affinity DataEC50:  526nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518740(CHEMBL4444106)
Affinity DataEC50:  570nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518756(CHEMBL1546037)
Affinity DataEC50:  640nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518743(CHEMBL4441168)
Affinity DataEC50:  701nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518737(CHEMBL4515644)
Affinity DataEC50:  712nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518753(CHEMBL4461752)
Affinity DataEC50:  903nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518740(CHEMBL4444106)
Affinity DataEC50:  966nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518739(CHEMBL280106)
Affinity DataEC50:  1.01E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518747(CHEMBL4469858)
Affinity DataEC50:  1.19E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518743(CHEMBL4441168)
Affinity DataEC50:  1.43E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518742(CHEMBL4527494)
Affinity DataEC50:  1.71E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518747(CHEMBL4469858)
Affinity DataEC50:  1.99E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518746(CHEMBL4555548)
Affinity DataEC50:  2.13E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM76464(3,5-diphenyl-1-(phenylmethyl)-1,2,4-triazole | SMR...)
Affinity DataEC50:  2.18E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518748(CHEMBL4451751)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518745(CHEMBL4518983)
Affinity DataEC50:  2.24E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518757(CHEMBL4515184)
Affinity DataEC50:  2.29E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518753(CHEMBL4461752)
Affinity DataEC50:  2.37E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518738(CHEMBL1357461)
Affinity DataEC50:  2.47E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518758(CHEMBL4552379)
Affinity DataEC50:  2.47E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518760(CHEMBL4458758)
Affinity DataEC50:  2.57E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518738(CHEMBL1357461)
Affinity DataEC50:  2.64E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518737(CHEMBL4515644)
Affinity DataEC50:  5.03E+3nMAssay Description:Agonist activity at full length human LXRalpha expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518745(CHEMBL4518983)
Affinity DataEC50:  5.65E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518748(CHEMBL4451751)
Affinity DataEC50:  6.15E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Benha University

Curated by ChEMBL
LigandPNGBDBM50518746(CHEMBL4555548)
Affinity DataEC50:  6.71E+3nMAssay Description:Agonist activity at full length human LXRbeta expressed in HEK293 cells harboring LXRE-Luc promoter by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed