Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50007304
TargetAmine oxidase [flavin-containing] B(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-2-phenylcyclopropanamine | cid_2723716 | (...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cells using beetle luciferin as substrate after 1 hr by MAO-Glo ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-2-phenylcyclopropanamine | cid_2723716 | (...)
Affinity DataIC50: 85nMAssay Description:Inhibition of recombinant human MAOA expressed in baculovirus infected BTI insect cells using beetle luciferin as substrate after 1 hr by MAO-Glo ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508345(CHEMBL4448235)
Affinity DataIC50: 210nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-2-phenylcyclopropanamine | cid_2723716 | (...)
Affinity DataIC50: 4.64E+3nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508351(CHEMBL4559695)
Affinity DataIC50: 7.58E+3nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508343(CHEMBL4588414)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508347(CHEMBL4448010)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508346(CHEMBL4475757)
Affinity DataIC50: 5.14E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508342(CHEMBL4437242)
Affinity DataIC50: 5.88E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508349(CHEMBL4470558)
Affinity DataIC50: 6.64E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508348(CHEMBL4465177)
Affinity DataIC50: 7.75E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508350(CHEMBL4442428)
Affinity DataIC50: 8.83E+4nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508344(CHEMBL4472145)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged LSD1 isoform2 (158 to end residues) expressed in Escherichia coli using methylated peptide as substrate pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508345(CHEMBL4448235)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human MAOB expressed in baculovirus infected BTI insect cells using beetle luciferin as substrate after 1 hr by MAO-Glo ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Taizhou People'S Hospital

Curated by ChEMBL
LigandPNGBDBM50508345(CHEMBL4448235)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of recombinant human MAOA expressed in baculovirus infected BTI insect cells using beetle luciferin as substrate after 1 hr by MAO-Glo ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed