Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008671
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521238(CHEMBL4589937)
Affinity DataEC50:  0.00640nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521239(CHEMBL4443026)
Affinity DataEC50:  0.0114nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521240(CHEMBL4535601)
Affinity DataEC50:  0.0139nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521241(CHEMBL4456936)
Affinity DataEC50:  0.00920nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521242(CHEMBL4456488)
Affinity DataEC50:  0.0103nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521243(CHEMBL4532868)
Affinity DataEC50:  0.00590nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521244(CHEMBL4525398)
Affinity DataEC50:  0.0117nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50521245(CHEMBL4547187)
Affinity DataEC50:  0.0130nMAssay Description:Inhibition of gamma-secretase (unknown origin) assessed as decrease in amyloid beta-42 secretion by cell based AlphaLisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed