Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50008677
TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521261(CHEMBL4584670)
Affinity DataEC50:  12nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521257(CHEMBL4537090)
Affinity DataEC50:  57nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521259(CHEMBL4592996)
Affinity DataEC50:  82nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521262(CHEMBL4464856)
Affinity DataEC50:  324nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521260(CHEMBL4573031)
Affinity DataEC50:  458nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50521258(CHEMBL4531290)
Affinity DataEC50:  4.92E+3nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as intracellular cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed