Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50010281
TargetSomatostatin receptor type 1(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  310nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataEC50:  2.30nMAssay Description:Binding affinity to human SSTR2 expressed in CHO-K1 cells assessed as induction of SSTR2 internalization after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  9.60nMAssay Description:Displacement of [125I]somatostatin from human SSTR5 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.290nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  20nMAssay Description:Displacement of [125I]somatostatin from human SSTR3 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataEC50:  1nMAssay Description:Binding affinity to human SSTR2 expressed in CHO-K1 cells assessed as induction of SSTR2 internalization after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.320nMAssay Description:Displacement of [125I]somatostatin from human SSTR5 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.200nMAssay Description:Displacement of [125I]somatostatin from human SSTR4 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  5.48E+3nMAssay Description:Displacement of [125I]somatostatin from human SSTR4 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.0320nMAssay Description:Displacement of [125I]somatostatin from human SSTR3 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537060(CHEMBL4575530)
Affinity DataEC50:  11nMAssay Description:Binding affinity to human SSTR2 expressed in CHO-K1 cells assessed as induction of SSTR2 internalization after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKi:  0.00500nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537063(CHEMBL4590517)
Affinity DataKi:  0.0130nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537069(CHEMBL4584764)
Affinity DataKi:  0.0150nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537077(CHEMBL4550617)
Affinity DataKi:  0.0150nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537066(CHEMBL4541310)
Affinity DataKi:  0.0150nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537076(CHEMBL4564727)
Affinity DataKi:  0.0180nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKi:  0.0220nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537068(CHEMBL4592483)
Affinity DataKi:  0.0610nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537070(CHEMBL4581874)
Affinity DataKi:  0.0750nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537074(CHEMBL4556000)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537062(CHEMBL4549303)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537067(CHEMBL4532058)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537075(CHEMBL4548228)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537064(CHEMBL4563111)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537071(CHEMBL4581646)
Affinity DataKi:  0.180nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537065(CHEMBL4537192)
Affinity DataKi:  0.190nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537078(CHEMBL4577466)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537073(CHEMBL4534477)
Affinity DataKi:  0.770nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537060(CHEMBL4575530)
Affinity DataKi:  0.970nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Tarveda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50537079(CHEMBL4587303)
Affinity DataKi:  3.35E+3nMAssay Description:Displacement of [125I]somatostatin from human SSTR2 expressed in CHO-K1 cell membranes after 240 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed