Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50009225
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50328731(Edoxaban | CHEMBL1269025)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526346(CHEMBL4526357)
Affinity DataIC50: 220nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526351(CHEMBL4561623)
Affinity DataIC50: 960nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526347(CHEMBL4474248)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50465842(Kirenol)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526355(CHEMBL4555342)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526354(CHEMBL4452613)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526356(CHEMBL4577469)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526352(CHEMBL4581081)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526348(CHEMBL4455162)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526349(CHEMBL4560959)
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526353(CHEMBL4464490)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50526350(CHEMBL4468511)
Affinity DataIC50: 2.79E+4nMAssay Description:Inhibition of human factor Xa using Z-D-Arg-Gly-Arg-pNA.2HCl as substrate preincubated for 15 mins followed by substrate addition by UV absorption an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed