Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50008889
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM50523327(CHEMBL4437198)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM50435003(ENDOXIFEN)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM50523326(CHEMBL4568316)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM50523329(CHEMBL4474808)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM50523330(CHEMBL4453737)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAromatase(Human)
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)

Curated by ChEMBL
LigandPNGBDBM50523328(CHEMBL1991089)
Affinity DataIC50: 9.53E+4nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed