Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50010314
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50355501(RUXOLITINIB PHOSPHATE | INCB-018424 | RUXOLITINIB ...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human JAK2 (828 to 1132 residues) expressed in baculovirus infected Sf9 insect cells using EQEDEPEGDYFEWLE as substrate after 1 hr by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50355501(RUXOLITINIB PHOSPHATE | INCB-018424 | RUXOLITINIB ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human JAK1 (837 to 1142 residues) expressed in baculovirus infected Sf9 insect cells using EQEDEPEGDYFEWLE as substrate after 1 hr by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM185700(US9271981, 1a | US9161939, 1a | US10875847, Compou...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant JAK1 (852 to 1142 residues) by Z-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM185700(US9271981, 1a | US9161939, 1a | US10875847, Compou...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant JAK2 (808 to 1132 residues) by Z-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537335(CHEMBL4559204)
Affinity DataIC50: 23nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537350(CHEMBL4555943)
Affinity DataIC50: 28nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537332(CHEMBL4552462)
Affinity DataIC50: 38nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537349(CHEMBL4574380)
Affinity DataIC50: 101nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537344(CHEMBL4540569)
Affinity DataIC50: 126nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537335(CHEMBL4559204)
Affinity DataIC50: 151nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537342(CHEMBL4525213)
Affinity DataIC50: 411nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537332(CHEMBL4552462)
Affinity DataIC50: 414nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM63961(SMR000499034 | 2-chloranyl-N-(1H-indazol-5-yl)benz...)
Affinity DataIC50: 453nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537350(CHEMBL4555943)
Affinity DataIC50: 460nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537329(CHEMBL4527179)
Affinity DataIC50: 583nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537340(CHEMBL4594048)
Affinity DataIC50: 718nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537340(CHEMBL4594048)
Affinity DataIC50: 764nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537337(CHEMBL4483633)
Affinity DataIC50: 820nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537329(CHEMBL4527179)
Affinity DataIC50: 943nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537342(CHEMBL4525213)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537339(CHEMBL4545256)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537346(CHEMBL4579262)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537349(CHEMBL4574380)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537336(CHEMBL4541350)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537328(CHEMBL4593760)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537344(CHEMBL4540569)
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537341(CHEMBL4541296)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537333(CHEMBL4585646)
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537343(CHEMBL4514766)
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537338(CHEMBL4572055)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537328(CHEMBL4593760)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537330(CHEMBL4514375)
Affinity DataIC50: 3.54E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537334(CHEMBL4569041)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537347(CHEMBL4532227)
Affinity DataIC50: 6.34E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537339(CHEMBL4545256)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM63961(SMR000499034 | 2-chloranyl-N-(1H-indazol-5-yl)benz...)
Affinity DataIC50: 8.53E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537345(CHEMBL4593750)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537338(CHEMBL4572055)
Affinity DataIC50: 9.29E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537345(CHEMBL4593750)
Affinity DataIC50: 9.53E+3nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537330(CHEMBL4514375)
Affinity DataIC50: 9.67E+3nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537333(CHEMBL4585646)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537343(CHEMBL4514766)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537337(CHEMBL4483633)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537331(CHEMBL1595400)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537351(CHEMBL4553196)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of JAK2 (unknown origin) after 1 hr FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537346(CHEMBL4579262)
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537336(CHEMBL4541350)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537334(CHEMBL4569041)
Affinity DataIC50: 2.41E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537341(CHEMBL4541296)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50537347(CHEMBL4532227)
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of JAK1 (unknown origin) after 1 hr by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
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