Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50008902
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: 4.74E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: 7.56E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: 8.54E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: 8.95E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: 9.41E+3nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523409(CHEMBL4483725)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523406(CHEMBL4536433)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin IV [1-448](malaria parasite P. falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 4 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523415(CHEMBL4515188)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin 2 using EDANS-CO-CH2-CH2-CO-ALERMFLSFP-Dap(DABCYL)OH as substrate measured after 60 mins by fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523412(CHEMBL4567098)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523410(CHEMBL4453475)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523408(CHEMBL4435264)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged BACE1 using Mca-SEVNLDAEFRK(Dpn)RR-NH2 as substrate measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523411(CHEMBL4475207)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523414(CHEMBL4436020)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523407(CHEMBL4438229)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Saint Louis University

Curated by ChEMBL
LigandPNGBDBM50523413(CHEMBL4576672)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Tracer Red binding to human ERG expressed in membranes by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed