Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50008961
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  0.0200nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  0.0300nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM50523980(CHEMBL4456753)
Affinity DataEC50:  1.20nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation incubated for 24 hrs in presence of 100 uM H2O2 by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM50523980(CHEMBL4456753)
Affinity DataEC50:  6.10nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation incubated for 24 hrs in presence of 50 uM H2O2 by luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM50523980(CHEMBL4456753)
Affinity DataEC50:  470nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM50106635(CHEMBL334773 | (+/-)-2,3-bis(4-hydroxyphenyl)propa...)
Affinity DataEC50:  7.20E+5nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation incubated for 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
University of Richmond

Curated by ChEMBL
LigandPNGBDBM50106635(CHEMBL334773 | (+/-)-2,3-bis(4-hydroxyphenyl)propa...)
Affinity DataEC50:  8.90E+5nMAssay Description:Activation of human ERbeta assessed as induction of transcriptional activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)