Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50008996
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 245nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 363nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 95nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 5.29E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 5.18E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 1.29E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 78nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 2.14E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 5.25E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 891nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 1.39E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 2.12E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 250nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 5.37E+3nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H2 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataEC50: 880nMAssay Description:Agonist activity at recombinant human Gs-coupled H2 receptor expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulat...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [I125]bolton hunter-CCK-8S from recombinant human CCK1 receptor expressed in stable CHO cells measured after 1 to 2 hrs by microscint...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 245nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of tracer Red binding to human ERG expressed in membranes after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 912nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.69E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.71E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.93E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 3.09E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 4.45E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 4.47E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 4.57E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Human)
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Academy of Scientific and Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 4.61E+3nMAssay Description:Antagonist activity at recombinant human Gi-coupled H3 receptor expressed in HEK293T cells assessed as reduction in histamine-induced inhibition of f...More data for this Ligand-Target Pair
