Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50011257
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546012(CHEMBL4761929)
Affinity DataEC50:  1.31E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546011(CHEMBL4741659)
Affinity DataEC50:  2.24E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546010(CHEMBL4750599)
Affinity DataEC50: <3.10E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546009(CHEMBL4750436)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546008(CHEMBL4784090)
Affinity DataEC50:  1.37E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546007(CHEMBL4795261)
Affinity DataEC50:  4.60E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546006(CHEMBL4747514)
Affinity DataEC50:  2.02E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546005(CHEMBL4758530)
Affinity DataEC50:  1.65E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546004(CHEMBL4759521)
Affinity DataEC50:  6.10E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546003(CHEMBL4759642)
Affinity DataEC50:  5.90E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546002(CHEMBL4747631)
Affinity DataEC50:  4.30E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546001(CHEMBL4776102)
Affinity DataEC50:  3.80E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546000(CHEMBL4780579)
Affinity DataEC50:  4.40E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50545999(CHEMBL4778307)
Affinity DataEC50:  9.50E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50545998(CHEMBL4745050)
Affinity DataEC50:  1.28E+4nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50197060(CHEMBL1417584)
Affinity DataEC50:  5.20E+3nMAssay Description:Activation of human TREK1 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50197060(CHEMBL1417584)
Affinity DataEC50:  7.70E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546011(CHEMBL4741659)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546010(CHEMBL4750599)
Affinity DataEC50: <3.60E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546009(CHEMBL4750436)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546008(CHEMBL4784090)
Affinity DataEC50:  2.65E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546007(CHEMBL4795261)
Affinity DataEC50:  5.60E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546006(CHEMBL4747514)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546005(CHEMBL4758530)
Affinity DataEC50:  2.85E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546004(CHEMBL4759521)
Affinity DataEC50:  5.50E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546003(CHEMBL4759642)
Affinity DataEC50:  7.70E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546002(CHEMBL4747631)
Affinity DataEC50:  5.90E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546001(CHEMBL4776102)
Affinity DataEC50:  6.80E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50546000(CHEMBL4780579)
Affinity DataEC50:  7.50E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50545999(CHEMBL4778307)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPotassium channel subfamily K member 10(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50545998(CHEMBL4745050)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of human TREK2 by thallium flux mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed