Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50009069
TargetAlbumin(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataKd:  99nMAssay Description:Displacement of dansylated phenylalanine from human serum albumin by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAlbumin(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataKd:  230nMAssay Description:Displacement of dansylated arginine from human serum albumin by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 3(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) using aggregate form of compound by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 3(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50011360(CHEMBL3260990)
Affinity DataKd:  2.00E+4nMAssay Description:Inhibition of 8-NBD-cAMP binding to human EPAC1 cAMP binding domain (149 to 318 residues) by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 3(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50280395(CHEMBL4171480)
Affinity DataKd:  1.24E+5nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetRap guanine nucleotide exchange factor 3(Human)
University Health Network

Curated by ChEMBL
LigandPNGBDBM50280395(CHEMBL4171480)
Affinity DataKd:  7.57E+5nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) in presence of human serum albumin by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed