Compile Data Set for Download or QSAR
Report error Found 144 Enz. Inhib. hit(s) with all data for entry = 50008157
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516264(CHEMBL4463013)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516261(CHEMBL4466640)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516249(CHEMBL4524602)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516262(CHEMBL4567690)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516238(CHEMBL4578966)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516250(CHEMBL4450173)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516237(CHEMBL4533562)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516260(CHEMBL4534007)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516251(CHEMBL4449377)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516256(CHEMBL4555599)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516257(CHEMBL4519913)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516242(CHEMBL4535004)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516253(CHEMBL4454168)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516246(CHEMBL4453295)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516252(CHEMBL4590515)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516239(CHEMBL4462028)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516265(CHEMBL4438188)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516244(CHEMBL4532150)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516236(CHEMBL4473591)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516240(CHEMBL4443398)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516245(CHEMBL4452900)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516243(CHEMBL4450343)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516254(CHEMBL4436064)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516235(CHEMBL4563408)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516258(CHEMBL4570109)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516255(CHEMBL4552147)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516259(CHEMBL4521215)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516247(CHEMBL4440543)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516248(CHEMBL4464256)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516260(CHEMBL4534007)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516241(CHEMBL4554452)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516250(CHEMBL4450173)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516261(CHEMBL4466640)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516249(CHEMBL4524602)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516235(CHEMBL4563408)
Affinity DataEC50:  718nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in CHOK1 cells co-expressing Galphaq16 assessed as reduction in CP55940-induced intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516263(CHEMBL4471789)
Affinity DataKi:  730nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516265(CHEMBL4438188)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516236(CHEMBL4473591)
Affinity DataEC50:  765nMAssay Description:Inverse agonist activity at human CB1 receptor expressed in CHOK1 cells co-expressing Galphaq16 assessed as reduction in CP55940-induced intracellula...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516240(CHEMBL4443398)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516264(CHEMBL4463013)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516238(CHEMBL4578966)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516254(CHEMBL4436064)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516237(CHEMBL4533562)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516258(CHEMBL4570109)
Affinity DataKi:  6.50E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516253(CHEMBL4454168)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516262(CHEMBL4567690)
Affinity DataKi:  7.60E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516235(CHEMBL4563408)
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of [3H]nisoxetine from recombinant human norepinephrine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516236(CHEMBL4473591)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]astemizole from human ERG measured after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516235(CHEMBL4563408)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]DADLE from recombinant human DOR after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50516235(CHEMBL4563408)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I](+/-)DOI from recombinant human 5HT2A receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
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