Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50008040
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes assessed as dissociation constant by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKd: 6.5nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes assessed as dissociation rate constant at 10 uM by liquid scintillation anal...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at MOR in Wistar rat brain membranes after 60 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Agonist activity at CB1R/CB2R in Wistar rat brain membranes after 60 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 134nMAssay Description:Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataEC50: 154nMAssay Description:Agonist activity at MOR in Wistar rat brain membranes after 60 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 172nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 183nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 186nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Displacement of [3H]WIN-55,212-2 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 214nMAssay Description:Displacement of [3H]Ile5,6-deltorphin-2 from DOR in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 231nMAssay Description:Displacement of [3H]HS-665 from KOR in guinea pig brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 247nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Centre of The Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 251nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes after 60 mins by liquid scintillation analysisMore data for this Ligand-Target Pair






















